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Pharmacokinetic and pharmacodynamic characteristics of ganirelix (Antagon/Orgalutran∗). part I. absolute bioavailability of 0.25 mg of ganirelix after.

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Presentation on theme: "Pharmacokinetic and pharmacodynamic characteristics of ganirelix (Antagon/Orgalutran∗). part I. absolute bioavailability of 0.25 mg of ganirelix after."— Presentation transcript:

1 Pharmacokinetic and pharmacodynamic characteristics of ganirelix (Antagon/Orgalutran∗). part I. absolute bioavailability of 0.25 mg of ganirelix after a single subcutaneous injection in healthy female volunteers  Janine J.L Oberyé, Bernadette M.J.L Mannaerts, Huub-Jan Kleijn, B.Sc., Cees J Timmer  Fertility and Sterility  Volume 72, Issue 6, Pages (December 1999) DOI: /S (99)

2 Figure 1 Log-linear plot of serum ganirelix concentrations after SC administration and IV administration of 0.25 mg of ganirelix to 15 healthy female volunteers. Oberyé. Ganirelix (Antagon/Orgalutran). Fertil Steril 1999. Fertility and Sterility  , DOI: ( /S (99) )

3 Figure 2 Systolic and diastolic blood pressure after SC administration (n = 18) and IV administration (n = 17) of 0.25 mg of ganirelix to healthy female volunteers. ▴ = systolic (IV); ▵ = systolic (SC); • = diastolic (IV); ○ = diastolic (SC). Oberyé. Ganirelix (Antagon/Orgalutran). Fertil Steril 1999. Fertility and Sterility  , DOI: ( /S (99) )


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