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2003-2004 Antineoplastics 1 February 2016 3:08 AM.

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Presentation on theme: "2003-2004 Antineoplastics 1 February 2016 3:08 AM."— Presentation transcript:

1 2003-2004 Antineoplastics 1 February 2016 3:08 AM

2 Alemtuzumab Antineoplastic Anti-CD52 antibody

3 Aminoglutethimide Antineoplastic Immunosuppressive Glucocorticoid antagonist Aromatase inhibitor (decreases steroid synthesis)

4 Amsacrine Antineoplastic Miscellaneous

5 Anastrozole Antineoplastic Antiestrogen Aromatase inhibitor

6 L-asparaginase Antineoplastic Protein synthesis inhibitor

7 Azathioprine Immunosuppressive Antineoplastic Antimetabolite (“pseudofeedback inhibition” of HGPRT and PRP)

8 Bleomycin Antineoplastic Natural product Antibiotic

9 Busulfan Antineoplastic Alkylating Agent

10 Carmustine (BCNU) Antineoplastic Alkylating Agent

11 Cisplatin Antineoplastic Miscellaneous Cross-linking agent

12 Cyclophosphamide Antineoplastic Alkylating Agent

13 Cyclosporine Immunosuppressive Antineoplastic Binds cyclophilin Inhibits calcineurin

14 Cyproterone acetate Antiandrogen Antineoplastic androgen receptor antagonist

15 Cytarabine (AraC) Antineoplastic Antimetabolite

16 Dacarbazine Antineoplastic Alkylating Agent

17 Dactinomycin Antineoplastic Natural product Antibiotic

18 Daunorubicin Antineoplastic Anthracycline antibiotic Natural product

19 Dexamethasone Adrenocorticosteroid Glucocorticoid Antineoplastic Anti-inflammatory steroid Not by inhalation

20 Doxorubicin Antineoplastic Anthracycline antibiotic Natural product

21 Etoposide Antineoplastic Natural product Plant alkaloid

22 Exemestane Antineoplastic Antiestrogen Aromatase Inhibitor

23 5-Fluorouracil Antineoplastic Antimetabolite Thymidylate synthase inhibitor

24 Fulvestrant Antineoplastic Antiestrogen Estrogen receptor antagonist

25 Gemtuzumab Antineoplastic Anti-CD33 antibody

26 Goserelin Antineoplastic Gonadotropin releasing hormone (GnRH) agonist

27 Hydroxyurea Antineoplastic Miscellaneous Ribonucleotide reductase inhibitor

28 Ibritumomab Antineoplastic Anti-CD20 antibody

29 Imatinib Antineoplastic Miscellaneous Tyrosine kinase inhibitor

30 Interleukin 2 Cytokine Antineoplastic

31 Interleukin 11 Cytokine Antineoplastic (supporting agent)

32 Iressa Antineoplastic Miscellaneous Tyrosine kinase inhibitor

33 Letrozole Antineoplastic Antiestrogen Aromatase Inhibitor

34 Leucovorin Antineoplastic (supporting agent) Folic acid analogue (used in methotrexate rescue)

35 Leuprolide Antineoplastic Gonadotropin releasing hormone (GnRH) agonist

36 Lomustine (CCNU) Antineoplastic Alkylating Agent

37 Mechlorethamine Antineoplastic Alkylating Agent

38 Melphalan Antineoplastic Alkylating Agent

39 6-Mercaptopurine Antineoplastic Antimetabolite (“pseudofeedback inhibition” of HGPRT and PRP – purine synthesis)

40 Mesna Antineoplastic (supporting agent) Prevent hemorrhagic cystitis due to cyclophosphamide

41 Methotrexate Immunosuppressive Antineoplastic Folic acid antagonist Dihydrofolate reductase inhibitor

42 Mitomycin C Antineoplastic Natural product Antibiotic

43 Paclitaxel Antineoplastic Natural product Plant alkaloid (taxane)

44 Pentostatin Antineoplastic Miscellaneous Enzyme inhibitor (blocks purine synthesis)

45 Rituxumab Antineoplastic Anti-CD20 antibody

46 Tacrolimus Immunosuppressive Antineoplastic Binds FKBP (FK506 binding protein) Inhibits calcineurin

47 Thalidomide Antineoplastic Anti-angiogenic Anti-TNF  Leprosy (not antibiotic)

48 6-Thioguanine Antineoplastic Antimetabolite (“pseudofeedback inhibition” of HGPRT and PRP – purine synthesis)

49 Thiotepa Antineoplastic Alkylating agent

50 Trastuzumab Antineoplastic Anti-HER2 antibody

51 Tumor necrosis factor  Cytokine Antineoplastic

52 Vinblastine Antineoplastic Vinca alkaloid Natural product

53 Vincristine Antineoplastic Vinca alkaloid Natural product


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