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Membrane Membrane receptors. Single-pass membrane receptors membrane.

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Presentation on theme: "Membrane Membrane receptors. Single-pass membrane receptors membrane."— Presentation transcript:

1 membrane Membrane receptors

2 Single-pass membrane receptors membrane

3 Multi-pass membrane receptors

4 Ion channel membrane receptors membrane + +

5 Ion channel membrane receptors

6 Receptor kinases

7 Kinase activities associated with receptors intrinsic tyrosine kinase activity JAK tyrosine kinase activity

8 G-protein-linked receptors GTP hormone membrane

9 G-protein-linked receptors    GDP

10 G-protein-linked receptors   adapter adenylate cyclase 

11 Insulin activation of glucose response IRS-1 P P PP P P GLUT

12 Follicle Stimulating Hormone & Receptor

13 FSH subunit mRNAs Huhtaniemi and Aittomaki (1998) Eur.J.Endo. 138: 473– 481

14 FSH subunit polypeptides Huhtaniemi and Aittomaki (1998) Eur.J.Endo. 138: 473– 481

15 FSH Fox, et al. Mol Endocrinol (2001) 15:378-389

16 FSH Receptor Huhtaniemi and Aittomaki (1998) Eur.J.Endo. 138: 473– 481 mRNA

17 FSH Receptor Huhtaniemi and Aittomaki (1998) Eur.J.Endo. 138: 473– 481

18 FSH Receptor (C, cysteine; S, serine; K, lysine; R, arginine; N, asparagine; A, alanine; D, aspartic acid; F, phenylalanine). Mann, et al. (2000) Biol. Reprod. 62: 1240-1247

19 FSH Receptor Mann, et al. (2000) Biol. Reprod. 62: 1240-1247

20 FSH Receptor Sohn, et al. (2003) J. Biol. Chem. 278: 47868 –47876

21 FSH Receptor Sohn, et al. (2003) J. Biol. Chem. 278: 47868 –47876

22 FSH Receptor Gay et al. (2006) Nature Reviews Immunology 6: 693-698

23 Natural mutations of FSH & Receptor Huhtaniemi and Aittomaki (1998) Eur.J.Endo. 138: 473– 481


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